Molecule Details
InChIKeyDMFLXIRKHPTWEU-UHFFFAOYSA-N
Compound Name1-(3-(tert-Butyl)-1-(p-tolyl)-1H-pyrazol-5-yl)-3-(4-((2-((3-methoxy-5-(3-morpholino-propoxy)phenyl)amino)pyrimidin-4-yl)oxy)naphthalen-1-yl)urea
Canonical SMILESCOc1cc(Nc2nccc(Oc3ccc(NC(=O)Nc4cc(C(C)(C)C)nn4-c4ccc(C)cc4)c4ccccc34)n2)cc(OCCCN2CCOCC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.37
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43405 SYK Homo sapiens Human PF07714 PF00017 7.7 IC50 ChEMBL;BindingDB
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 7.6 IC50 ChEMBL;BindingDB
P53778 MAPK12 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB