Molecule Details
InChIKeyDLFSESWOWKXVMD-UHFFFAOYSA-N
Compound NameN-[5-(1,1-dioxo-1lambda*6*-isothiazolidin-2-yl)-1H-indazol-3-yl]-2-m-tolyl-acetamide
Canonical SMILESCc1cccc(CC(=O)Nc2n[nH]c3ccc(N4CCCS4(=O)=O)cc23)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.77
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 8.0 pIC50 TTD_MultiTarget
P06493 CDK1 Homo sapiens Human PF00069 7.7 pIC50 TTD_MultiTarget
P11802 CDK4 Homo sapiens Human PF00069 7.7 pIC50 TTD_MultiTarget