Molecule Details
InChIKeyDLDXMINZRQNSDI-CQSZACIVSA-N
Compound Name6-N-(3-amino-5-chlorophenyl)-2-N-[(3R)-piperidin-3-yl]-9-propan-2-ylpurine-2,6-diamine
Canonical SMILESCC(C)n1cnc2c(Nc3cc(N)cc(Cl)c3)nc(N[C@@H]3CCCNC3)nc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49760 CLK2 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P49759 CLK1 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
Q9HAZ1 CLK4 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB