Molecule Details
InChIKeyDLCOOKRUECVLCI-UHFFFAOYSA-N
Compound NameN~2~-(1h-Benzimidazol-6-Yl)-N~4~-(5-Cyclobutyl-1h-Pyrazol-3-Yl)quinazoline-2,4-Diamine
Canonical SMILESc1ccc2c(Nc3cc(C4CCC4)[nH]n3)nc(Nc3ccc4[nH]cnc4c3)nc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75385 ULK1 Homo sapiens Human PF12063 PF21127 PF00069 8.1 IC50 ChEMBL;BindingDB
Q8IYT8 ULK2 Homo sapiens Human PF12063 PF21127 PF00069 7.9 IC50 ChEMBL;BindingDB
Q15118 PDK1 Homo sapiens Human PF10436 PF02518 6.4 IC50 ChEMBL;BindingDB