Molecule Details
InChIKeyDKHFDFCYFZTWRU-UHFFFAOYSA-N
Canonical SMILESCOc1cc(OC)c(F)c(N2Cc3cnc(-c4cn(C)nc4C)cc3N(C3CC(=O)N(C)C3)C2=O)c1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P21802 FGFR2 Homo sapiens Human PF07679 PF13927 PF07714 6.9 IC50 ChEMBL;BindingDB
P22607 FGFR3 Homo sapiens Human PF21165 PF07679 PF13927 PF07714 6.9 IC50 ChEMBL;BindingDB