Molecule Details
InChIKeyDKDNNTGJSLIDOQ-UHFFFAOYSA-N
Compound NameN-(5-Sulfamoyl-[1,3,4]thiadiazol-2-yl)-3-trifluoromethanesulfonylamino-propionamide
Canonical SMILESNS(=O)(=O)c1nnc(NC(=O)CCNS(=O)(=O)C(F)(F)F)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.89
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.9 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.9 pIC50 TTD_MultiTarget