Molecule Details
InChIKeyDJVTZQIKKLGURV-APWZRJJASA-N
Compound Name(R)-2-({4-[((R)-2-Amino-3-mercapto-propylamino)-methyl]-biphenyl-2-carbonyl}-amino)-3-methylsulfanyl-propionic acid
Canonical SMILESCSC[C@H](NC(=O)c1cc(CNC[C@@H](N)CS)ccc1-c1ccccc1)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.63
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.3 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.3 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 7.3 IC50 ChEMBL