Molecule Details
InChIKeyDINLHKGZVRGQQO-UHFFFAOYSA-N
Compound Name1-Methyl-4-[(1-spiro[2.5]octan-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]pyrrole-2-carboxamide
Canonical SMILESCn1cc(Nc2ncc3cnn(C4CCC5(CC4)CC5)c3n2)cc1C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
P06493 CDK1 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB