Molecule Details
InChIKeyDIKKTLPJDURHSW-UHFFFAOYSA-N
Compound Name2-methyl-N-((1-(4-phenylpiperazin-1-yl)cyclohexyl)methyl)-1,2,3,4-tetrahydroisoquinoline-5-carboxamide
Canonical SMILESCN1CCc2c(cccc2C(=O)NCC2(N3CCN(c4ccccc4)CC3)CCCCC2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.8 Ki ChEMBL
Q99572 P2RX7 Homo sapiens Human PF20478 PF00864 7.5 IC50 ChEMBL
Q01959 SLC6A3 Homo sapiens Human PF00209 6.5 IC50 ChEMBL;BindingDB