Molecule Details
InChIKeyDIFGLRSYVDIDJS-JHOUSYSJSA-N
Compound NameUS8598206, Table 6, 7
Canonical SMILESN=C(N)c1ccc(CNC(=O)[C@H](CCC2CCNCC2)NC(=O)[C@@H](CCC2CCN(C(=O)C3CC3)CC2)NS(=O)(=O)Cc2ccccc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 9.5 Ki ChEMBL;BindingDB
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 9.2 Ki ChEMBL;BindingDB
P03951 F11 Homo sapiens Human PF00024 PF00089 6.2 Ki ChEMBL;BindingDB