Molecule Details
InChIKeyDHXMASVOPVPEJZ-QRKDJJKOSA-N
Canonical SMILESNC(N)=NCCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H](N)CCCN=C(N)N)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.85
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30411 BDKRB2 Homo sapiens Human PF00001 7.8 pIC50 TTD_MultiTarget
P46663 BDKRB1 Homo sapiens Human PF00001 7.8 pIC50 TTD_MultiTarget