Molecule Details
InChIKeyDHXAFRBSJGTAFK-UHFFFAOYSA-N
Compound Name6-Acetyl-2-[[5-[4-(2-chloroacetyl)piperazin-1-yl]-2-pyridinyl]amino]-8-cyclopentyl-5-methylpyrido[2,3-d]pyrimidin-7-one
Canonical SMILESCC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCl)CC4)cn3)nc2n(C2CCCC2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.03
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P30281 CCND3 Homo sapiens Human PF02984 PF00134 8.0 IC50 ChEMBL
Q00534 CDK6 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB