Molecule Details
InChIKeyDHXAAEUVXXASMB-UHFFFAOYSA-N
Compound Name2-(3-(1-(Phenylsulfonyl)cyclobutyl)propyl)-1,2,3,4-tetrahydroisoquinoline
Canonical SMILESO=S(=O)(c1ccccc1)C1(CCCN2CCc3ccccc3C2)CCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P34969 HTR7 Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB