Molecule Details
InChIKeyDHUULRFMFRMVOC-JZPFNFMMSA-N
Compound Name(S)-2-[2-({(S)-3-Methyl-2-[2-(3-pyridin-4-ylmethyl-3H-imidazol-4-yl)-acetylamino]-pentyl}-naphthalen-1-ylmethyl-amino)-acetylamino]-4-methylsulfanyl-butyric acid
Canonical SMILESCCC(C)[C@@H](CN(CC(=O)N[C@@H](CCSC)C(=O)O)Cc1cccc2ccccc12)NC(=O)Cc1cncn1Cc1ccncc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.55
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.6 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.6 IC50 ChEMBL