Molecule Details
InChIKeyDGYXXVVLRDGURB-UHFFFAOYSA-N
Canonical SMILESCC(C)N(CC(N)=O)C(=O)c1cc2c(N(C)C)nc(NCCc3c[nH]c4ccccc34)nc2n1CCCc1ccc(Cl)cc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O15151 MDM4 Homo sapiens Human PF13920 PF00641 6.2 Ki ChEMBL;BindingDB
Q00987 MDM2 Homo sapiens Human PF02201 PF13920 PF00641 6.2 Ki ChEMBL;BindingDB