Molecule Details
InChIKeyDGXYDPJRLWCWFV-ZXDVGYGBSA-N
Compound Name2,2-Dimethyl-propionic acid (3R,3aS)-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazol-7-yl ester
Canonical SMILESC/C(=C\c1ccccc1)CN1CCN(C[C@@H]2ON=C3c4ccc(OC(=O)C(C)(C)C)cc4OC[C@H]32)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18825 ADRA2C Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.9 Ki ChEMBL;BindingDB