Molecule Details
InChIKeyDGTSSSGHGKXRIS-UHFFFAOYSA-N
Compound Name4-[[[3-[(4-Cyanophenyl)methyl]imidazol-4-yl]methyl-methylamino]methyl]-3-(3-ethoxyphenyl)benzonitrile
Canonical SMILESCCOc1cccc(-c2cc(C#N)ccc2CN(C)Cc2cncn2Cc2ccc(C#N)cc2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL10.52
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 10.5 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 10.5 IC50 ChEMBL;BindingDB