Molecule Details
InChIKeyDGLDUQZIRFLLRH-QVWWMRLHSA-N
Compound Name(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-benzyl-1-(3,4-dichlorophenyl)-N-methylcyclopropanecarboxamide
Canonical SMILESCC(=O)NC1(c2ccccc2)CCN(C[C@@H]2C[C@@]2(C(=O)N(C)Cc2ccccc2)c2ccc(Cl)c(Cl)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29371 TACR3 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P21452 TACR2 Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB
P25103 TACR1 Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB