Molecule Details
InChIKeyDGISRQRHSYAYQM-UHFFFAOYSA-N
Compound Name2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-N-(4-{2-[3-(2-amino-ethyl)-1H-indol-5-yloxy]-acetylamino}-phenyl)-acetamide
Canonical SMILESNCCc1c[nH]c2ccc(OCC(=O)Nc3ccc(NC(=O)COc4ccc5[nH]cc(CCN)c5c4)cc3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 10.0 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 9.6 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB