Molecule Details
InChIKeyDFXFMJLXQWVGCL-UHFFFAOYSA-N
Compound Name5-[5-Amino-7-(4-nuorophenyl)-2-[(1,3-thiazol-2-yl)methyl]-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-1-methyl-1,2-dihydropyridin-2-one
Canonical SMILESCn1cc(-c2c(-c3ccc(F)cc3)nc(N)n3nc(Cc4nccs4)nc23)ccc1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.66
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 8.1 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB