Molecule Details
InChIKeyDFOCUWZXJBAUSQ-URLMMPGGSA-N
Compound Name(+)-Berbamine
Canonical SMILESCOc1cc2c3cc1Oc1c(OC)c(OC)cc4c1[C@@H](Cc1ccc(O)c(c1)Oc1ccc(cc1)C[C@@H]3N(C)CC2)N(C)CC4
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.36
SourceChEMBL
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB18146
Drug NameBerbamine
CAS Number478-61-5
Groups experimental
ATC Codes nan
Descriptionnan

Categories: Alkaloids Analgesics Analgesics, Non-Narcotic Anti-Inflammatory Agents Anti-Inflammatory Agents, Non-Steroidal Antiarrhythmic agents Antihypertensive Agents Antirheumatic Agents Calcium Channel Blockers Calcium-Regulating Hormones and Agents Cardiovascular Agents Heterocyclic Compounds, Fused-Ring Isoquinolines Membrane Transport Modulators Peripheral Nervous System Agents Sensory System Agents
Cross-references: BindingDB: 50241654 ChEBI: 3063 CHEMBL504323 ChemSpider: 242126 C09357 Wikipedia: Berbamine ZINC: ZINC000030726840
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9H2S1 KCNN2 Homo sapiens Human PF02888 PF07885 PF03530 6.5 Ki ChEMBL
Q9UGI6 KCNN3 Homo sapiens Human PF02888 PF07885 PF03530 6.2 Ki ChEMBL