Molecule Details
InChIKeyDFINWNNMGCBCLX-YIUPACBUSA-N
Canonical SMILESC[C@@H](NC(=O)N1CCC(NC(=O)c2nccs2)CC1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](Cc1ccccc1)C(=O)[C@@]1(C)CO1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.41
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P28062 PSMB8 Homo sapiens Human PF00227 6.5 IC50 ChEMBL;BindingDB
P28074 PSMB5 Homo sapiens Human PF00227 6.3 IC50 ChEMBL;BindingDB