Molecule Details
InChIKeyDFBYFJSXUCUKLA-UHFFFAOYSA-N
Compound Name5-[5-(3,4,5-trimethoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyridin-2-amine
Canonical SMILESCOc1cc(-c2cnc3[nH]cc(-c4ccc(N)nc4)c3c2)cc(OC)c1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5S007 LRRK2 Homo sapiens Human PF23745 PF23744 PF23748 PF16095 PF25497 PF13855 PF00069 PF08477 8.3 IC50 ChEMBL;BindingDB
Q16584 MAP3K11 Homo sapiens Human PF07714 PF14604 8.2 IC50 ChEMBL;BindingDB