Molecule Details
InChIKeyDEPFXQSAHGKYPV-UHFFFAOYSA-N
Compound Name2-[[5-Chloro-2-(4-methoxyphenoxy)pyrimidin-4-yl]amino]benzamide
Canonical SMILESCOc1ccc(Oc2ncc(Cl)c(Nc3ccccc3C(N)=O)n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.28
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB