Molecule Details
InChIKeyDDVHSMTXNFZEQH-LHLGERLTSA-N
Compound Name(2S,3S,4S,5R,6S)-3,4,5-Trihydroxy-6-{4-[(4-sulfamoyl-benzoylamino)-methyl]-[1,2,3]triazol-1-yloxy}-tetrahydro-pyran-2-carboxylic acid methyl ester
Canonical SMILESCOC(=O)[C@H]1O[C@@H](On2cc(CNC(=O)c3ccc(S(N)(=O)=O)cc3)nn2)[C@H](O)[C@@H](O)[C@@H]1O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.83
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 7.6 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.4 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.4 pIC50 TTD_MultiTarget