Molecule Details
InChIKeyDDNOBRYGXQJOJB-UHFFFAOYSA-N
Compound Name5-[4-(Heptadecafluorooctylsulfonylamino)phenylsulfonylamino]-1,3,4-thiadiazole-2-sulfonamide
Canonical SMILESNS(=O)(=O)c1nnc(NS(=O)(=O)c2ccc(NS(=O)(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)cc2)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.83
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.7 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.7 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 6.1 Ki ChEMBL;BindingDB