InChIKey	DDLIGBOFAVUZHB-UHFFFAOYSA-N
Compound Name	Midazolam
Canonical SMILES	Cc1ncc2n1-c1ccc(Cl)cc1C(c1ccccc1F)=NC2
Clinical Status	Data-mined Candidate
Targets (Human+Pathogen)	3
Pfam Stratification	Cross-Family
Avg pChEMBL	7.21
Source	BindingDB;ChEMBL

DrugBank ID	DB00683
Drug Name	Midazolam
CAS Number	59467-70-8
Groups	approved illicit investigational
ATC Codes	N05CD08
Description	Midazolam is a short-acting hypnotic-sedative drug with anxiolytic, muscle relaxant, anticonvulsant, sedative, hypnotic, and amnesic properties.[A173842] It belongs to a class of drugs called _benzodiazepines_. This drug is unique from others in this class due to its rapid onset of effects and short...

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Categories: Adjuvants, Anesthesia Anesthetics Anti-Anxiety Agents Benzodiazepine hypnotics and sedatives Benzodiazepines and benzodiazepine derivatives Central Nervous System Agents Central Nervous System Depressants Cytochrome P-450 CYP3A Inhibitors Cytochrome P-450 CYP3A Substrates Cytochrome P-450 CYP3A4 Inhibitors Cytochrome P-450 CYP3A4 Inhibitors (strength unknown) Cytochrome P-450 CYP3A4 Substrates Cytochrome P-450 CYP3A5 Substrates Cytochrome P-450 CYP3A7 Substrates Cytochrome P-450 Enzyme Inhibitors Cytochrome P-450 Substrates Drugs that are Mainly Renally Excreted GABA Agents GABA Modulators Heterocyclic Compounds, Fused-Ring Hypnotics and Sedatives Nervous System Neurotransmitter Agents P-glycoprotein substrates Psycholeptics Psychotropic Drugs Tranquilizing Agents Triazolobenzodiazepines UGT1A4 substrates UGT2B7 substrates

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Cross-references: BindingDB: 21363 ChEBI: 6931 CHEMBL655 ChemSpider: 4047 Drugs Product Database (DPD): 11188 Guide to Pharmacology: 3342 IUPHAR: 3342 C07524 D00550 PDB: 08J PharmGKB: PA450496 PubChem:4192 PubChem:46507611 RxCUI: 6960 Therapeutic Targets Database: DAP000241 Wikipedia: Midazolam ZINC: ZINC000095626706