Molecule Details
InChIKeyDDKIKSYBXRUQAD-UHFFFAOYSA-N
Canonical SMILESCOc1ccc(-n2nc(C(C)(C)C)cc2NC(=O)Nc2ccc(Oc3cc(Nc4cc(OC)cc(C(=O)NCCN5CCOCC5)c4)ncn3)c3ccccc23)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.4 IC50 ChEMBL;BindingDB
P49840 GSK3A Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB