Molecule Details
InChIKeyDDCGYKUGMMDSDD-UHFFFAOYSA-N
Compound Name1-(2-Phenyl-3H-imidazol-4-ylmethyl)-4-pyridin-3-yl-piperazine
Canonical SMILESc1ccc(-c2nc(CN3CCN(c4cccnc4)CC3)c[nH]2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB