Molecule Details
InChIKeyDCUODGWOKBGFJV-NYPGBQQYSA-N
Compound Name(14Z,21S)-21-benzyl-8,26-dichloro-12,17-dioxa-1,4,19,22,24-pentaazatricyclo[21.3.1.0^{6,11}]heptacosa-6(11),7,9,14,23,25-hexaene-3,18,27-trione
Canonical SMILESO=C1Cn2c(Cl)cnc(c2=O)N[C@@H](Cc2ccccc2)CNC(=O)OC/C=C\COc2ccc(Cl)cc2CN1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.47
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 10.2 Ki ChEMBL;BindingDB
P00750 PLAT Homo sapiens Human PF00008 PF00039 PF00051 PF00089 8.2 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 7.0 Ki ChEMBL;BindingDB