Molecule Details
InChIKeyDCLSJFXDVAAQJQ-GERZZCHPSA-N
Canonical SMILESCc1ncc(-c2c(C#N)ccc(Cl)c2F)nc1C(=O)Nc1cnn(C(C)c2cnc(N3C[C@H]4C[C@H]4C3=O)c(F)c2C)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.96
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 9.7 IC50 ChEMBL;BindingDB
P03951 F11 Homo sapiens Human PF00024 PF00089 6.2 IC50 BindingDB