Molecule Details
InChIKeyDCIBEKBKAOZGMO-UHFFFAOYSA-N
Compound NameN-[1-Allyl-3-(toluene-4-sulfonyl)-1H-pyrrolo[2,3-b]quinoxalin-2-yl]-benzenesulfonamide
Canonical SMILESC=CCn1c(NS(=O)(=O)c2ccccc2)c(S(=O)(=O)c2ccc(C)cc2)c2nc3ccccc3nc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.18
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBE0 SAE1 Homo sapiens Human PF00899 6.3 IC50 ChEMBL;BindingDB
Q9UBT2 UBA2 Homo sapiens Human PF00899 PF14732 PF16195 6.2 IC50 ChEMBL
P63279 UBE2I Homo sapiens Human PF00179 6.1 IC50 BindingDB