Molecule Details
InChIKeyDCHWBJNKHKXUAM-UHFFFAOYSA-N
Compound Name3-[[2-[carbamimidoyl(methyl)amino]acetyl]amino]-N-(5-sulfamoyl-1,3,4-thiadiazol-2-yl)propanamide
Canonical SMILESCN(CC(=O)NCCC(=O)Nc1nnc(S(N)(=O)=O)s1)C(=N)N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.36
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.7 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.7 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.7 Ki ChEMBL;BindingDB