Molecule Details
InChIKeyDCHQNZAIUFIFEB-UHFFFAOYSA-N
Compound Name6-[2-(dimethylamino)ethyl]-N-[5-fluoro-4-(7-fluoro-2,3-dimethylbenzimidazol-5-yl)pyrimidin-2-yl]-7,8-dihydro-5H-1,6-naphthyridin-2-amine
Canonical SMILESCc1nc2c(F)cc(-c3nc(Nc4ccc5c(n4)CCN(CCN(C)C)C5)ncc3F)cc2n1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P30281 CCND3 Homo sapiens Human PF02984 PF00134 7.9 IC50 ChEMBL
Q00534 CDK6 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB