Molecule Details
InChIKeyDBRBZVDPIWOVAV-RJISSDALSA-N
Compound NameH-Ala-Leu-Cys(1)-Asn-Cys(2)-Asn-D-Arg-Ile-Ile-Ile-Pro-His-Met-Cys(1)-Trp-Lys-Lys-Cys(2)-Gly-Lys-Lys-NH2
Canonical SMILESCC[C@H](C)[C@@H]1NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@@H](CCCNC(=N)N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]2CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)N)C(=O)N[C@@H](CC(N)=O)C(=O)N2)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@@H]2CCCN2C(=O)[C@H]([C@@H](C)CC)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P48048 KCNJ1 Homo sapiens Human PF01007 PF17655 8.7 Ki ChEMBL;BindingDB
P48544 KCNJ5 Homo sapiens Human PF01007 PF17655 8.1 Ki ChEMBL;BindingDB
P48549 KCNJ3 Homo sapiens Human PF01007 PF17655 8.1 Ki ChEMBL