Molecule Details
InChIKeyDBQMDBXMFKWIGE-OAQYLSRUSA-N
Compound Name4-[(3R)-3-benzyl-4-(4-sulfamoylbenzoyl)piperazine-1-carbonyl]benzenesulfonamide
Canonical SMILESNS(=O)(=O)c1ccc(C(=O)N2CCN(C(=O)c3ccc(S(N)(=O)=O)cc3)[C@H](Cc3ccccc3)C2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P22748 CA4 Homo sapiens Human PF00194 8.3 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 8.1 Ki ChEMBL;BindingDB
P00915 CA1 Homo sapiens Human PF00194 7.2 Ki ChEMBL;BindingDB