Molecule Details
InChIKeyDBLYNSSCIKMVDW-WUFINQPMSA-N
Compound Name(7S,10R)-10-(benzylsulfonylamino)-N-[(4-carbamimidoylphenyl)methyl]-4,9,13-trioxo-3,8,14-triazabicyclo[14.3.1]icosa-1(19),16(20),17-triene-7-carboxamide
Canonical SMILESN=C(N)c1ccc(CNC(=O)[C@@H]2CCC(=O)NCc3cccc(c3)CNC(=O)CC[C@@H](NS(=O)(=O)Cc3ccccc3)C(=O)N2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P04070 PROC Homo sapiens Human PF14670 PF00594 PF00089 8.3 Ki ChEMBL;BindingDB
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 7.6 Ki ChEMBL;BindingDB
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 6.4 Ki ChEMBL;BindingDB