Molecule Details
InChIKeyDBFVYHGYASQAJI-UHFFFAOYSA-N
Compound Name3-amino-N-[4-[3-(aminomethyl)piperidin-1-yl]-3-pyridinyl]pyrazine-2-carboxamide
Canonical SMILESNCC1CCCN(c2ccncc2NC(=O)c2nccnc2N)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.14
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.0 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 7.3 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.2 Ki ChEMBL;BindingDB