Molecule Details
InChIKeyDAKWJOSEOVIBIL-UHFFFAOYSA-N
Compound Name3-(6-amino-3-pyridinyl)-6-piperidin-4-ylsulfinyl-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESNc1ccc(-c2ccc([S+]([O-])C3CCNCC3)c(S(N)(=O)=O)c2-c2nn[nH]n2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.08
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 8.5 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 8.2 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 7.6 IC50 BindingDB