Molecule Details
InChIKeyDADQHECQKQBHAW-UHFFFAOYSA-N
Compound NameN,N-diisopentyl-2-(4-(methylcarbamoyl)phenylamino)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide
Canonical SMILESCNC(=O)c1ccc(Nc2nc3ccc(C(=O)N(CCC(C)C)CCC(C)C)cc3n2CCCN2CCCCC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.14
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB