Molecule Details
InChIKeyDACGDZLVWJQELB-UHFFFAOYSA-N
Compound Name2-[carbamimidoyl(methyl)amino]-N-[4-[(5-sulfamoyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl]acetamide
Canonical SMILESCN(CC(=O)Nc1ccc(S(=O)(=O)Nc2nnc(S(N)(=O)=O)s2)cc1)C(=N)N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.61
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 9.0 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 9.0 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.9 Ki ChEMBL;BindingDB