Molecule Details
InChIKeyDAAGOCSHXCDWDY-ZDUSSCGKSA-N
Compound Name3-(1,3-Benzodioxol-5-yl)-N-[(1S)-1-phenylethyl]-isoxazolo[5,4-c]pyridin-5-amine
Canonical SMILESC[C@H](Nc1cc2c(-c3ccc4c(c3)OCO4)noc2cn1)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NYY3 PLK2 Homo sapiens Human PF00069 PF00659 8.4 IC50 ChEMBL;BindingDB
Q9H4B4 PLK3 Homo sapiens Human PF00069 PF00659 7.6 IC50 ChEMBL;BindingDB
P53350 PLK1 Homo sapiens Human PF00069 PF00659 6.7 IC50 ChEMBL;BindingDB