Molecule Details
InChIKeyCZOGJFVDQVTTBG-LBPRGKRZSA-N
Compound Name4-amino-2-(furan-2-yl)-6-[(2S)-2-hydroxypropoxy]-N-[(3-methyl-2-pyridinyl)methyl]pyrimidine-5-carboxamide
Canonical SMILESCc1cccnc1CNC(=O)c1c(N)nc(-c2ccco2)nc1OC[C@H](C)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 8.5 IC50 ChEMBL;BindingDB
P0DMS8 ADORA3 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB