Molecule Details
InChIKeyCZMFKHZKGYYFSP-UHFFFAOYSA-N
Compound Name7-cyclopentyl-N-(2-fluorophenyl)-2-[(5-piperazin-1-yl-2-pyridinyl)amino]pyrrolo[2,3-d]pyrimidine-6-carboxamide
Canonical SMILESO=C(Nc1ccccc1F)c1cc2cnc(Nc3ccc(N4CCNCC4)cn3)nc2n1C1CCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
P24385 CCND1 Homo sapiens Human PF02984 PF00134 6.4 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 6.4 IC50 ChEMBL