Molecule Details
InChIKeyCZLALGVBUDRCJM-FWEHEUNISA-N
Compound NameN-[(S)-1-((S)-1-{(S)-1-[(S)-1-Carbamoyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-4-guanidino-butylcarbamoyl}-2-phenyl-ethylcarbamoyl)-2-(3H-imidazol-4-yl)-ethyl]-oxalamide
Canonical SMILESN=C(N)NCCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)C(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01726 MC1R Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB