Molecule Details
InChIKeyCZCBVFVSSWZKPW-UHFFFAOYSA-N
Compound Name4-methyl-N-[3-methyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl]-3-(2-pyrazolo[1,5-a]pyrimidin-6-ylethynyl)benzamide
Canonical SMILESCc1cc(CN2CCN(C)CC2)cc(NC(=O)c2ccc(C)c(C#Cc3cnc4ccnn4c3)c2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q08345 DDR1 Homo sapiens Human PF21114 PF00754 PF07714 8.2 IC50 ChEMBL;BindingDB
Q16832 DDR2 Homo sapiens Human PF21114 PF00754 PF07714 7.4 IC50 ChEMBL;BindingDB
P10721 KIT Homo sapiens Human PF00047 PF07714 6.6 IC50 ChEMBL;BindingDB