Molecule Details
InChIKeyCYUNIDFFVZCUDT-UHFFFAOYSA-N
Compound Name8-[4-(Cyclopropylmethyl)piperazin-1-yl]-3-thia-1,7-diazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaene
Canonical SMILESc1cc2c(N3CCN(CC4CC4)CC3)nc3ccsc3n2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.5 IC50 ChEMBL;BindingDB