Molecule Details
InChIKeyCYRMEVWUFYIIFZ-UHFFFAOYSA-N
Compound Name3-(3-methyl-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl)-2-(1H-tetrazol-5-yl)-6-trifluoromethyl)benzenesulfonamide
Canonical SMILESCc1n[nH]c2c1CN(c1ccc(C(F)(F)F)c(S(N)(=O)=O)c1-c1nnn[nH]1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.92
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 9.7 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.0 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.1 IC50 BindingDB