Molecule Details
InChIKeyCYOQMLSODZDBGH-UHFFFAOYSA-N
Compound Name1-[6-(1,4-diazepan-1-yl)-2-pyridinyl]-6-(1H-pyrazol-4-yl)pyrazolo[4,3-c]pyridine
Canonical SMILESc1cc(N2CCCNCC2)nc(-n2ncc3cnc(-c4cn[nH]c4)cc32)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 10.1 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.9 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.8 Ki ChEMBL;BindingDB