Molecule Details
InChIKeyCYMDODRBHNOOOT-UHFFFAOYSA-N
Compound Name3-{4-[5-(2,5-Dimethyl-pyrrolidin-1-yl)-pentyl]-3-oxo-3,4-dihydro-2H-benzo[1,4]oxazin-2-yl}-benzamidine
Canonical SMILESCC1CCC(C)N1CCCCCN1C(=O)C(c2cccc(C(=N)N)c2)Oc2ccccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.3 IC50 ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 6.1 IC50 ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.0 IC50 ChEMBL;BindingDB